A First-in-Class, Highly Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 6
Yudao Shen,Fengling Li,Magdalena M. Szewczyk,Levon Halabelian,Irene Chau,Mohammad S. Eram,Carlo Dela Sena,Kwang-Su Park,Fanye Meng,He Chen,Hong Zeng,Aiping Dong,Hong Wu,Viacheslav V. Trush,David McLeod,Carlos A. Zepeda-Velazquez,Robert M. Campbell,Mary M. Mader,Brian M. Watson,Matthieu Schapira,Cheryl H. Arrowsmith,Rima Al-Awar,Dalia Barsyte-Lovejoy,H. Umit Kaniskan,Peter J. Brown,Masoud Vedadi,Jian Jin JOURNAL OF MEDICINAL CHEMISTRY(2021)
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