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Orally Bioavailable and Site-Selective Covalent STING Inhibitor Derived from a Macrocyclic Marine Diterpenoid.

Guang-Hao Niu,Wan-Chi Hsiao, Po-Hsun Lee, Li-Guo Zheng, Yu-Shao Yang, Wei-Cheng Huang,Chih-Chien Hsieh,Tai-Yu Chiu, Jing-Ya Wang,Ching-Ping Chen,Chen-Lung Huang, May-Su You, Yi-Ping Kuo, Chien-Ming Wang,Zhi-Hong Wen,Guann-Yi Yu,Chiung-Tong Chen,Ya-Hui Chi,Chun-Wei Tung, Shu-Ching Hsu,Teng-Kuang Yeh,Ping-Jyun Sung,Mingzi M Zhang,Lun Kelvin Tsou

Journal of medicinal chemistry(2025)

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