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Disrupted Target Binding with Acryloyl Group As Potential Bcr-Abl/C-Src Dual Kinase Inhibitor Optimization Strategies with Maintained Antitumor Activity

Ching Lin, Hsin-Yi Chiang,Grace Shiahuy Chen,Ji-Wang Chern,Chao-Wu Yu

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS(2025)

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关键词
Kinase inhibitor,Anticancer,Acryloyl group,Quinolone
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