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Computational-aided Rational Mutation Design of Pertuzumab to Overcome Active HER2 Mutation S310F Through Antibody-Drug Conjugates.

Xuefei Bai,Lingyi Xu,Zhe Wang,Xinlei Zhuang, Jiangtao Ning, Yanping Sun, Haibin Wang, Yugang Guo,Yingchun Xu,Jiangtao Guo,Shuqing Chen,Liqiang Pan

PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA(2025)

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关键词
antibody engineering,directed evolution,drug resistance
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