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The Discovery of MORF-627, a Highly Selective Conformationally-Biased Zwitterionic Integrin Αvβ6 Inhibitor for Fibrosis

Bryce A. Harrison,James E. Dowling,Matthew G. Bursavich,Dawn M. Troast, Katherine M. Chong, Kristopher N. Hahn,Cheng Zhong, Kristen M. Mulvihill, Hanh Nguyen, Meghan F. Monroy,Qi Qiao, Brian Sosa,Siavash Mostafavi, Inese Smukste,Dooyoung Lee,Laura Cappellucci, Elizabeth H. Konopka, Patrycja Nowakowski,Lukasz Stawski, Mayra Senices, Minh Hai Nguyen, Parmita S. Kapoor,Lia Luus,Andrew Sullivan, Andrea Bortolato, Mats Svensson, Eugene R. Hickey, Kyle D. Konze,Tyler Day, Byungchan Kim, Ana Negri,Aleksey I. Gerasyuto,Terence I. Moy,Min Lu,Adrian S. Ray,Liangsu Wang,Dan Cui,Fu-Yang Lin,Blaise Lippa,Bruce N. Rogers

JOURNAL OF MEDICINAL CHEMISTRY(2024)

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