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Synthesis and Biological Evaluation of Ortho-Phenyl Phenylhydroxamic Acids Containing Phenothiazine with Improved Selectivity for Class IIa Histone Deacetylases

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY(2024)

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关键词
Class IIa histone deacetylases (HDACs),structure-activity relationship (SAR),molecular modelling,cancer cells
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