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Enhanced Radiotheranostic Targeting of Integrin Α5β1 with PEGylation-enabled Peptide Multidisplay Platform (pegibody): A Strategy for Prolonged Tumor Retention with Fast Blood Clearance

Siqi Zhang, Xiaohui Ma,Jiang Wu,Jieting Shen, Yuntao Shi,Xingkai Wang,Lin Xie,Xiaona Sun,Yuxuan Wu,Hao Tian, Xin Gao, Xueyao Chen, Hongyi Huang, Lu Chen, Xuekai Song, Qichen Hu,Hailong Zhang,Feng Wang,Zhao-Hui Jin,Ming-Rong Zhang

Acta Pharmaceutica Sinica B(2024)

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关键词
Integrin α5β1,Peptide,PET imaging,Targeted radionuclide therapy,PEGylation,Tumor,Multidisplay,PEGibody
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