Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido[2,3-d]pyrimidin-7-one-based SOS1 inhibitor

Kun Wang,Zehui Zhou, Xinyi Ma, Jiahang Xu, Wangyang Xu,Guizhen Zhou,Chuan Zhou, Huajie Li,Mingyue Zheng,Sulin Zhang,Tianfeng Xu

Bioorganic & Medicinal Chemistry Letters(2024)

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