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Discovery of a Novel Orally Bioavailable FLT3-PROTAC Degrader for Efficient Treatment of Acute Myeloid Leukemia and Overcoming Resistance of FLT3 Inhibitors

Junwei Wang,Quanjin Rong, Lei Ye,Bingqian Fang, Yifan Zhao, Yu Sun, Haikun Zhou,Dan Wang, Jinting He,Zhenzhen Cui, Qijian Zhang,Di Kang,Lihong Hu

JOURNAL OF MEDICINAL CHEMISTRY(2024)

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