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Discovery of First-in-class DOT1L Inhibitors Against the R231Q Gain-of-function Mutation in the Catalytic Domain with Therapeutic Potential of Lung Cancer

Acta Pharmaceutica Sinica B(2024)

引用 2|浏览20
关键词
DOT1L,R231Q mutation,Lung cancer,Adenosine-containing inhibitors,Epigenetics
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