Development of a Scalable Synthesis of the Small Molecule TGFβR1 Inhibitor BMS-986260
Muthalagu Vetrichelvan,Souvik Rakshit, Sathishkumar Chandrasekaran, Karthikeyan Chinnakalai,Chetan Padmakar Darne, Dyamanna Doddalingappa, Indasi Gopikumar,Anuradha Gupta,Arun Kumar Gupta,Ananta Karmakar,Thirumalai Lakshminarasimhan,David K. Leahy,Senthil Palani,Vignesh Radhakrishnan,Richard Rampulla,Antony Savarimuthu, Varadharajan Subramanian,Upender Velaparthi,Jayakumar Warrier,Martin D. Eastgate Organic Process Research & Development(2020)
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TGFβR1 inhibitor,imidazo[1,2-b]pyridazine,TosMIC,AKTS software,Van Leusen imidazole synthesis
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