Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead MSC-4106
Timo Heinrich, Carl Peterson,Richard Schneider,Sakshi Garg,Daniel Schwarz,Jakub Gunera,Anita Seshire,Lisa Kötzner,Sarah Schlesiger,Djordje Musil,Heike Schilke, Benjamin Doerfel, Patrizia Diehl, Pia Böpple,Ana R. Lemos,Pedro M. F. Sousa,Filipe Freire,Tiago M. Bandeiras,Emma Carswell, Nicholas Pearson, Sameer Sirohi, Mollie Hooker,Elisabeth Trivier, Rebecca Broome, Alexander Balsiger, Abigail Crowden,Christian Dillon,Dirk Wienke Journal of Medicinal Chemistry(2022)
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