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Toward the Development of a Manufacturing Process for Milvexian: Scale-Up Synthesis of the Side Chain

Simon Wagschal,Diego Broggini, Trung D. C. Cao,Pascal Schleiss,Kristian Paun, Jessica Steiner, Anna-Lena Merk,Joachim Harsdorf, Winfried Fiedler,Stefan Schirling, Sven Hock, Tobias Strittmatter,Jan Dijkmans,Ivan Vervest, Tim Van Hoegaerden, Brecht Egle,Matthew P. Mower,Zhi Liu, Zhiyong Cao, Xiaoning He, Lei Chen, Lei Qin, Hongyu Tan, Jun Yan,Nicolas Lucien Cuniere,Carolyn S. Wei,Venkata Vuyyuru,Rajaram Ayothiraman,Sundaramurthy Rangaswamy, Mohamed Jaleel,Rajappa Vaidyanathan,Martin D. Eastgate,Richard Klep,Cyril Benhaim,Ilse Vogels, Koen Peeters,Sebastien Lemaire

ORGANIC PROCESS RESEARCH & DEVELOPMENT(2023)

引用 2|浏览27
关键词
milvexian,Suzuki,click,azide,chlorination,factor XIa inhibitor
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