Discovery of a Potent and Orally Bioavailable Zwitterionic Series of Selective Estrogen Receptor Degrader-Antagonists
James S. Scott,Darren Stead,Bernard Barlaam,Jason Breed,Rodrigo J. Carbajo,Elisabetta Chiarparin,Natalie Cureton,Paul R. J. Davey,David I. Fisher,Eric T. Gangl,Tyler Grebe,Ryan D. Greenwood,Sudhir Hande,Holia Hatoum-Mokdad,Samantha J. Hughes,Thomas A. Hunt,Tony Johnson,Stefan L. Kavanagh,Teresa C. M. Klinowska,Carrie J. B. Larner,Mandy Lawson,Andrew S. Lister,David Longmire,Stacey Marden,Thomas M. McGuire, Caroline McMillan,Lindsay McMurray,Christopher J. Morrow,J. Willem M. Nissink,Thomas A. Moss,Daniel H. O'Donovan,Radoslaw Polanski,Stephen Stokes,Kumar Thakur,Dawn Trueman,Caroline Truman,Michael J. Tucker,Haixia Wang,Nicky Whalley,Dedong Wu,Ye Wu,Bin Yang,Wenzhan Yang JOURNAL OF MEDICINAL CHEMISTRY(2023)
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