Development of KT-253, a Highly Potent and Selective Heterobifunctional MDM2 Degrader for the Treatment of Acute Myeloid Leukemia
Michele Mayo,Yogesh Chutake,Rahul Karnik,Alice McDonald,Patricia S. Cho,Jessica Filiatrault,Dapeng Chen,Vaishali Dixit,William Proctor,Susanne Breitkopf, Frank Qi,Kan-Nian Hu,Kirti Sharma,Reggie Ewesuedo,Matt Weiss,Joseph D. Growney,Juliet Williams,Stefanie S. Schalm BLOOD(2022)
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