Cyclin dependent kinase 9 inhibition as a potential treatment for hepatocellular carcinoma

JOURNAL OF CLINICAL ONCOLOGY(2022)

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摘要
We demonstrated the in vitro and in vivo activity of CDK9 inhibition on multiple HCC cell lines. Our data support further clinical development of CDK9 inhibitors as a treatment for HCC.
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关键词
Apoptosis,Cell line,Cyclin,Cyclin-dependent kinase 9,Hepatocellular carcinoma,Myeloid cell leukemia-1,Orthotopic model,Preclinical study,RNA polymerase,Xenograft
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