(1S,2R,3S,4S,5R,6R)‐2‐アミノ‐3‐[(3,4‐ジフルオロフェニル)スルファニルメチル]‐4‐ヒドロキシ‐ビシクロ[3.1.0]ヘキサン‐2,6‐ジカルボン酸塩酸塩(LY3020371HCl)の発見: 抗鬱様活性を持つ強力な向代謝性グルタミン酸2/3受容体アンタゴニスト
D Chappell Mark,Renhua Li,C Smith Stephon,Alexander Bruce,G Tromiczak Eric,E Tripp Allie,Blanco Maria‐Jesus,V Glukhareva Tatiana,J Quimby Steven,M. A. James,C. B. Thomas,Matthias Adam,M Schkeryantz Jeffrey,Mayhugh Daniel,A Erickson Jon, Gertraud Mark,Jaramillo Carlos,Mercedes Carpintero,DE Diego Jose Eugenio,Mario Barberis,Susana Garcı́a-Cerrada,F Soriano Jose,A. Stephen,Atwell Shane,Macewan Iain,Condon Bradley,Sougias Christine,Wang Jing,Aiping Zhang,Conners Kris,Groshong Chris,Rosary Stephen,Williams John,M Witkin Jeffrey, Xueyan Cao,Overshiner Carl,A Wafford Keith,Seidel Wesley,Xu-Shan Wang,A Heinz Beverly,Swanson Steven,Tudor John,W Bedwell David,Amber M. James,H Mitch Charles,L Ornstein Paul Journal of Medicinal Chemistry(2016)
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