(1S,2R,3S,4S,5R,6R)‐2‐アミノ‐3‐[(3,4‐ジフルオロフェニル)スルファニルメチル]‐4‐ヒドロキシ‐ビシクロ[3.1.0]ヘキサン‐2,6‐ジカルボン酸塩酸塩(LY3020371HCl)の発見: 抗鬱様活性を持つ強力な向代謝性グルタミン酸2/3受容体アンタゴニスト

D Chappell Mark,LI Renhua, C Smith Stephon, A Dressman Bruce, G Tromiczak Eric, E Tripp Allie,Blanco Maria‐Jesus, Vetman Tatiana, J Quimby Steven, Matthew T. James, C Britton Thomas, M Fivush Adam, M Schkeryantz Jeffrey, Mayhugh Daniel, A Erickson Jon, G Bures Mark,Jaramillo Carlos, Carpintero Mercedes, DE Diego Jose Eugenio,Barberis Mario, Garcia‐Cerrada Susana, F Soriano Jose,Antonysamy Stephen,Atwell Shane,Macewan Iain,Condon Bradley, Sougias Christine, Wang Jing,Zhang Aiping, Conners Kris,Groshong Chris, R Wasserman Stephen, W Koss John, M Witkin Jeffrey,Li Xia, Overshiner Carl, A Wafford Keith, Seidel Wesley,Wang Xu‐Shan, A Heinz Beverly,Swanson Steven, T Catlow John, W Bedwell David, A Monn James, H Mitch Charles, L Ornstein Paul

Journal of Medicinal Chemistry(2016)

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