非人類霊長類での中央部Aβを低減するイミノ複素環系β‐位アミロイド前駆体蛋白質切断酵素(BACE)阻害剤の構造ベース設計

Mandal Mihirbaran,WU Yusheng, Misiaszek Jeffrey,LI Guoqing,Buevich Alexei, P Caldwell John,Liu Xiaoxiang, D Mazzola Robert,Orth Peter,Strickland Corey,Voigt Johannes,Wang Hongwu,Zhu Zhaoning,Chen Xia,Grzelak Michael, A Hyde Lynn,Kuvelkar Reshma, T Leach Prescott,Terracina Giuseppe,Zhang Lili, Zhang Qi, S Michener Maria, Smith Brad,Cox Kathleen,Grotz Diane,Favreau Leonard,Mitra Kaushik,Kazakevich Irina, A Mckittrick Brian,Greenlee William, E Kennedy Matthew, M Parker Eric, N Cumming Jared, W Stamford Andrew

Journal of Medicinal Chemistry(2016)

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