Synthesis, Optimization, and Large-Scale Preparation of the Low-Dose Central Nervous System-Penetrant BACE1 Inhibitor LY3202626 via a [3 + 2] Nitrone Cycloaddition

Organic Process Research & Development(2020)

引用 6|浏览6
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关键词
BACE inhibitor,thermal nitrone cyclization,classical resolution,thiazine formation
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