From Protein To Candidate: Discovery Of Epz-5676, A Potent And Selective Inhibitor Of The Histone Methyltransferase Dot1l
Richard Chesworth,Edward J. Olhava,Kevin W. Kuntz,Aravind Basavapathruni,Christina R. A. Majer,Chris J. Sneeringer,Christina J. Allain,Alejandra Raimondi,Christine R. Klaus,Margaret Porter Scott,Carly A. Therkelsen,Scott R. Daigle,Roy M. Pollock,Victoria M. Richon,Robert A. Copeland,Ann Boriack-Sjodin,Lei Jin,Nigel J. Waters, Lee Arnold, Michael Patane,Paul Pearson, Joelle Sacks,Mikel P. Moyer ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY(2013)
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