In-Depth Characterization and Validation in BRG1-Mutant Lung Cancers Define Novel Catalytic Inhibitors of SWI/SNF Chromatin Remodeling
Zainab Jagani,Gregg Chenail,Kay Xiang,Geoffrey Bushold,Hyo-Eun C. Bhang,Ailing Li,GiNell Elliott,Jiang Zhu,Anthony Vattay,Tamara Gilbert,Anka Bric,Rie Kikkawa,Valérie Dubost,Rémi Terranova,John Cantwell,Catherine Luu,Serena Silver, Matt Shirley, Francois Huet,Rob Maher,John Reece-Hoyes,David Ruddy,Daniel Rakiec,Joshua Korn,Carsten Russ,Vera Ruda,Julia Dooley,Emily Costa,Isabel Park,Henrik Moebitz,Katsumasa Nakajima,Christopher D. Adair,Simon Mathieu,Rukundo Ntaganda,Troy Smith,David Farley,Daniel King,Xiaoling Xie,Raviraj Kulathila,Tiancen Hu,Xuewen Pan,Qicheng Ma,Katarina Vulic,Florencia Rago,Scott Clarkson,Robin Ge,Frederic Sigoillot,Gwynn Pardee,Linda Bagdasarian,Margaret McLaughlin,Kristy Haas,Jan Weiler,Steve Kovats,Mariela Jaskelioff, Marie Apolline-Gerard,Johanna Beil,Ulrike Naumann,Pascal Fortin,Frank P. Stegmeier,Michael G. Acker,Juliet Williams,Matthew Meyer,James E. Bradner,Nicholas Keen,William R. Sellers,Francesco Hofmann,Jeffrey A. Engelman,Darrin Stuart,Julien P.N. Papillon bioRxiv(2019)
Key words
SWI/SNF Complexes
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