Efficient Affinity Ranking of Fluorinated Ligands by 19F NMR: CSAR and FastCSAR
Journal of Biomolecular NMR(2020)
关键词
Fluorine NMR,Spin lock,Affinity ranking,Chemical shift anisotropy (CSA),Fragment-based drug design (FBDD),Density functional theory (DFT) calculations,Drug discovery
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