Discovery of 4-Arylquinoline-2-carboxamides, Highly Potent and Selective Class of Mglur2 Negative Allosteric Modulators: from HTS to Activity in Animal Models
Bioorganic & Medicinal Chemistry Letters(2020)
关键词
Metabotropic glutamate receptor 2,mGluR2 antagonists,High throughput screening,Cognition,Alzheimer’s disease
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