Abstract C036: Discovery of IACS-13909, an Allosteric SHP2 Inhibitor That Overcomes Multiple Mechanisms Underlying Osimertinib Resistance
Yuting Sun,Brooke A. Meyers,Sarah B. Johnson,Angela L. Harris,Barbara Czako,Jason B. Cross,Paul G. Leonard,Faika Mseeh,Maria E. Di Francesco,Connor A. Parker,Qi Wu,Christopher A. Bristow,Jason P. Burke,Caroline C. Carrillo,Christopher L. Carroll,Qing Chang,Ningping Feng,Sonal Gera,Gao Guang, Justin Kwang-Lay Huang,Yongying Jiang,Zhijun Kang,Jeffrey J. Kovacs,Xiaoyan Ma,Pijus K. Mandal,Timothy McAfoos,Robert A. Mullinax,Michael D. Peoples,Vandhana Ramamoorthy,Sahil Seth,Erika Suzuki, Christopher Conrad Williams,Simon S. Yu,Andy M. Zuniga,Giulio F. Draetta,Joseph R. Marszalek,Timothy P. Heffernan,Nancy E. Kohl,Philip Jones MOLECULAR CANCER THERAPEUTICS(2019)
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