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Abstract P1-10-08: Development of a First-in-class Oral Selective ERα Covalent Antagonist (SERCA) for the Treatment of ERαWT and ERαMUT Breast Cancer

M Korpal,X Puyang, C Furman,GZ Zheng,D Banka, J Wu,Z Zhang,M Thomas,C Mackenzie, H Yao,V Rimkunas,P Kumar,B Caleb, C Karr,V Subramanian, S Irwin,N Larsen,F Vaillancourt,T-V Nguyen, A Davis,B Chan,MH Hao, M O'Shea,S Prajapati,S Agoulnik, G Kuznetsov,N Kumar, Y Yu, G Lai, A Hart, S Eckley,P Fekkes, T Bowser,JJ Joshi,A Selvaraj,S Wardell, J Norris,S Smith, D Reynolds, L Mitchell,J Wang,L Yu,A Kim,N Rioux,T Sahmoud,M Warmuth,PG Smith,P Zhu

Cancer Research(2018)

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