Discovery of Selective Estrogen Receptor Covalent Antagonists for the Treatment of ER alphaWTand ER alphaMUTBreast Cancer.

X. Puyang, C. Furman,G.Z. Zheng,Z.J. Wu, D. Banka, K. Aithal,Sergei Agoulnik, D.M. Bolduc,S. Buonamici,B. Caleb,S. Das,Sean Eckley, P. Fekkes,M.H. Hao,Andrew Hart,René Houtman, S. Irwin, J.J. Joshi, C. Karr,A. Kim,Namita Kumar,P. Kumar,Galina Kuznetsov, W.G. Lai, N. Larsen, C. Mackenzie,Lesley-Ann Martin,Diana Melchers, A. Moriarty,T.V. Nguyen,John D. Norris, M. O'Shea, Sunil Pancholi, S. Prajapati, S. Rajagopalan, D.J. Reynolds, V. Rimkunas,N. Rioux,Ricardo Ribas,Amy Siu, S. Sivakumar,V. Subramanian, M. Thomas, F.H. Vaillancourt,J. Wang, Suzanne E. Wardell,M.J. Wick, S. Yao,L. Yu,M. Warmuth, P.G. Smith,P. Zhu,Manav Korpal

Cancer Discovery(2018)

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