General Methods for the Synthesis and Late-Stage Diversification of 2,4-Substituted 7-Azaindoles
Jeffrey G. Varnes,Thomas McGuire,Rebecca E. Meadows,Bernard Barlaam, Jemma Clark,Calum R. Cook, Gemma Davison,Allan Dishington,Chris De Savi,Craig Donald,Tyler Grebe,Sudhir Hande,Janet Hawkins,Alexander W. Hird,Jane Holmes,Andrew Lister,Simon Lucas,Jane Moore,Esther Moore,Anil Patel,Kurt G. Pike,Bryan Roberts,Andrew Stark,Darren Stead,Kumar Thakur,Paul Turner,Melissa Vasbinder,Bin Yang Tetrahedron Letters(2016)
关键词
7-Azaindole,Miyaura borylation,Suzuki-Miyaura reaction,1H-Pyrrolo[2,3-b]pyridine,2-(Piperidin-4-yl)-7-azaindole
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