Optimizing a Weakly Binding Fragment into a Potent RORγt Inverse Agonist with Efficacy in an in Vivo Inflammation Model.David A. Carcache,Anna Vulpetti,Joerg Kallen,Henri Mattes,David Orain,Rowan Stringer,Eric Vangrevelinghe,Romain M. Wolf,Klemens Kaupmann,Johannes Ottl,Janet Dawson,Nigel G. Cooke,Klemens Hoegenauer,Andreas Billich,Juergen Wagner,Christine Guntermann,Samuel HintermannJournal of Medicinal Chemistry(2018)引用 27|浏览51AI 理解论文溯源树样例生成溯源树,研究论文发展脉络Chat Paper正在生成论文摘要