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Synergistic Effect of Phosphorothioate, 5′-Vinylphosphonate and GalNAc Modifications for Enhancing Activity of Synthetic Sirna

Bioorganic & Medicinal Chemistry Letters(2016)

引用 42|浏览39
关键词
3 '-GalNAc cluster,5 '-Vinylphosphonate siRNA,Fully modified siRNA,Alternating F/OMe siRNA,siRNA phosphorothioates
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