Structure-Based Design of Orally Bioavailable 1H-Pyrrolo[3,2-c]pyridine Inhibitors of Mitotic Kinase Monopolar Spindle 1 (MPS1)
Sebastien Naud,Isaac M. Westwood,Amir Faisal,Peter Sheldrake,Vassilios Bavetsias,Butrus Atrash,Kwai-Ming J. Cheung,Manjuan Liu,Angela Hayes,Jessica Schmitt,Amy Wood,Vanessa Choi,Kathy Boxall,Grace Mak,Mark Gurden,Melanie Valenti,Alexis de Haven Brandon,Alan Henley,Ross Baker,Craig McAndrew,Berry Matijssen,Rosemary Burke,Swen Hoelder,Suzanne A. Eccles,Florence I. Raynaud,Spiros Linardopoulos,Rob L. M. van Montfort,Julian Blagg JOURNAL OF MEDICINAL CHEMISTRY(2013)
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Mitotic Checkpoint,Spindle Assembly
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