Estrogen receptor ligands. Part 6: Synthesis and binding affinity of dihydrobenzodithiins.

Bioorganic & Medicinal Chemistry Letters(2004)

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摘要
The synthesis and biological activity of dihydrobenzodithiins, as ERα-selective estrogen receptor ligands, are described.
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关键词
Estrogen receptor,Dihydrobenzodithiins,SERM,SERAM
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