Synthesis and in vitro DMPK profiling of a 1,2-dioxolane-based library with activity against Plasmodium falciparum

Bioorganic & Medicinal Chemistry Letters(2009)

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摘要
The synthesis, antiplasmodial activity and DMPK properties of a 43-member 1,2-dioxolane library is reported.
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关键词
Malaria,Antiplasmodial,1,2-Dioxolanes,DMPK profiling
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