Scaffold Oriented Synthesis. Part 4: Design, Synthesis and Biological Evaluation of Novel 5-Substituted Indazoles As Potent and Selective Kinase Inhibitors Employing Heterocycle Forming and Multicomponent Reactions
Bioorganic & medicinal chemistry letters(2011)
关键词
Kinase scaffolds,Kinase inhibitors,Gsk3 beta inhibitors,Rock2 inhibitors,Egfr inhibitors,Imidazopyrimidine,Imidazopyridines,Van Leusen reactions,MCR, multicomponent reactions
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