Selective androgen receptor modulators based on a series of 7H-[1,4]oxazino[3,2-g]quinolin-7-ones with improved in vivo activity
Bioorganic & Medicinal Chemistry Letters(2008)
摘要
The synthesis and biological evaluation of a selective androgen receptor modulator (SARM) with improved in vivo activity is reported.
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关键词
Androgen,SARM,Testosterone,Anabolic,Androgenic,Benzoxazine,AR,Muscle,Oxazino[3,2-g]quinolin-7-one
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