Substituted acyclic sulfonamides as human cannabinoid-1 receptor inverse agonists
Bioorganic & Medicinal Chemistry Letters, pp. 2184-2187, 2007.
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Keywords:
CannabinoidCB-1RSulfonamideObesity
Abstract:
Sulfonamide analogues of the potent CB1R inverse agonist 2 (Taranabant) were optimized for CB1R activity.
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