Thienopyridine urea inhibitors of KDR kinase
H. Robin Heyman,Robin R. Frey,Peter F. Bousquet,George A. Cunha,Maria D. Moskey,Asma A. Ahmed,Niru B. Soni,Patrick A. Marcotte,Lori J. Pease,Keith B. Glaser,Melinda Yates,Jennifer J. Bouska,Daniel H. Albert,Candace L. Black-Schaefer,Peter J. Dandliker,Kent D. Stewart,Paul Rafferty,Steven K. Davidsen,Michael R. Michaelides,Michael L. Curtin Bioorganic & Medicinal Chemistry Letters(2007)
摘要
The evaluation of KDR kinase inhibitor 2 (IC50=9nM) and related analogs is reported.
更多查看译文
关键词
KDR kinase,VEGF,Thienopyridine,Urea
AI 理解论文
溯源树
样例