Pyrazolopyridinones as functionally selective GABAA ligands
Bioorganic & Medicinal Chemistry Letters(2005)
摘要
2,5-Dihydro-3H-pyrazolo[4,3-c]pyridin-3-ones are GABAA receptor benzodiazepine binding site ligands, which can exhibit functional selectivity for the α3 subtype over the α1 subtype. SAR studies to optimize this functional selectivity are described.
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关键词
Pyrazolopyridinones,GABAA
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