Tricyclic thienopyridine–pyrimidones/thienopyrimidine–pyrimidones as orally efficacious mGluR1 antagonists for neuropathic pain
Bioorganic & Medicinal Chemistry Letters(2009)
摘要
A series of highly potent and selective mGluR1 antagonists have been discovered and demonstrated efficacy in animal model for pain.
更多查看译文
关键词
Tricyclic thienopyridine–pyrimidone,Thienopyrimidine–pyrimidone,Triazafluorenone,mGluR1 antagonist,Neuropathic pain
AI 理解论文
溯源树
样例
生成溯源树,研究论文发展脉络
Chat Paper
正在生成论文摘要