Design, synthesis and antibacterial activity of 3-methylenepyrrolidine formyl hydroxyamino derivatives as novel peptide deformylase inhibitors.

Bioorganic & Medicinal Chemistry Letters(2011)

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摘要
Design and synthesis of 3-methylenepyrrolidine formyl hydroxyamino derivatives as novel peptide deformylase inhibitors, and their antibacterial activities against susceptible and resistant clinical isolates including Gram-positive bacterial strains and Gram-negative ones have been reported.
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关键词
PDF inhibitor,Antibiotics,Drug-resistant bacteria,Pyrrolidine derivatives
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