Discovery of Potent, Soluble and Orally Active Trpv1 Antagonists. Structure-Activity Relationships of A Series of Isoxazoles
Paul Ratcliffe,Lynn Abernethy,Nasrin Ansari,Ken Cameron,Tom Clarkson,Maureen Dempster,David Dunn,Anna-Marie Easson,Darren Edwards,Katy Everett,Helen Feilden,Koc-Kan Ho,Steve Kultgen,Peter Littlewood,John Maclean,Duncan McArthur,Deborah McGregor,Hazel McLuskey,Irina Neagu,Olaf Nimz,Lesley-Anne Nisbet,Michael Ohlmeyer,Ronnie Palin,Quynhchi Pham,Yajing Rong,Andrew Roughton,Melanie Sammons,Robert Swanson,Heather Tracey,Glenn Walker Bioorganic & Medicinal Chemistry Letters(2011)
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TRPV1 antagonist,Antihyperalgesia,Isoxazoles
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