Verongamine, a Novel Bromotyrosine-Derived Histamine H3-Antagonist from the Marine Sponge Verongula gigantea

JOURNAL OF NATURAL PRODUCTS(1994)

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摘要
The novel bromotyrosine derivative verongamine [1] has been isolated from the marine sponge Verongula gigantea. The isolation of verongamine was facilitated by employing histamine-H-3 bioassay-guided fractionation. Verongamine is a specific histamine-H-3 antagonist at concentrations as low as 1 mu g/ml.
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关键词
verongamine,histamine,sponge,bromotyrosine-derived
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